Tolperisone
Muscle Relaxant · Skeletal muscle relaxant
Indications
Muscle spasm associated with locomotor diseases, neurological disorders, rehabilitation, peripheral vascular disorders.
Dosage
Tab: Adults: 150-450 mg 3 times daily. Children: 3 mth-6 yr, 5-10 mg/kg/day divided into 3 doses (1-3 tab daily); 6-14 yr, 4-2 mg/kg/day divided into 3 doses.
Adverse Effects
Muscular weakness, somnolence (rarely) in paediatrics.
Risk Factor (Pregnancy/Lactation)
Pregnancy: Contraindicated in pregnancy. Contraindications: Myasthaenia gravis.
Advice to Patient
Take with meals.
Pharmacokinetics
Absorption: Rapid. Metabolism: Hepatic. Bioavailability: 17%. Half-life elimination: 1.5-2.5 hrs. Time to peak, plasma: Oral: 0.5-1 hr. Excretion: Urine.
Brands with this active ingredient
Compiled by Healify Pharmacy from published drug references. How we compile it →
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