Tianeptine Sodium
Antidepressant · Presynaptic serotonin reuptake enhancer
Indications
Depression.
Dosage
Adults: 12.5 mg three times daily. Elderly: 25 mg daily. Children: Not recommended.
Adverse Effects
Epigastric pain, abdominal pain, dry mouth, anorexia, nausea, vomiting, constipation, flatulence, insomnia, drowsiness, nightmares, asthaenia, tachycardia, extrasystoles, pre-cordial pain, vertigo, headache, lipothymia, tremor, hot flushes, respiratory discomfort, lump in throat, myalgia, back pain.
Risk Factor (Pregnancy/Lactation)
Pregnancy: Contraindicated in pregnancy. Lactation: Contraindicated or not recommended. Precautions: See literature.
Interactions
MAOIs.
Advice to Patient
Take before main meals.
Pharmacokinetics
Absorption: Well absorbed. Metabolism: Extrarenal. Bioavailability: Approx. 99%. Half-life elimination: Approx. 2.5 hrs. Time to peak, plasma: Within 1 hr. Excretion: Urine. Faeces.
Compiled by Healify Pharmacy from published drug references. How we compile it →
Always consult a pharmacist or doctor.